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HM03
CAS No. 500565-15-1
HM03( —— )
Catalog No. M22402 CAS No. 500565-15-1
HM03 is a potent and selective inhibitor of HSPA5, and has anticancer activity.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 42 | Get Quote |
|
| 10MG | 72 | Get Quote |
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| 25MG | 140 | Get Quote |
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| 50MG | 258 | Get Quote |
|
| 100MG | 447 | Get Quote |
|
| 200MG | 584 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameHM03
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NoteResearch use only, not for human use.
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Brief DescriptionHM03 is a potent and selective inhibitor of HSPA5, and has anticancer activity.
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DescriptionHM03 is a potent and selective inhibitor of HSPA5, and has anticancer activity.
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In VitroCell Viability Assay Cell Line:HCT116 cells Concentration:0.1, 1, 10, 25, 50 μM Incubation Time:72 hours Result:Exhibited prominent inhibition effect (18% survival at 25 μM).
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In Vivo——
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Synonyms——
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PathwayCytoskeleton/Cell Adhesion Molecules
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TargetHSP
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RecptorHSPA5
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Research Area——
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Indication——
Chemical Information
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CAS Number500565-15-1
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Formula Weight462.97
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Molecular FormulaC26H27ClN4O2
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Purity>98% (HPLC)
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SolubilityDMSO:125 mg/mL (270.00 mM; Need ultrasonic)
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SMILESCOc1ccc2nc3cc(Cl)ccc3c(Nc3ccc(O)c(CN4CCN(C)CC4)c3)c2c1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Huang M , Li Z , Li D , et al. Structure-based design of HSPA5 inhibitors: From peptide to small molecule inhibitors[J]. Bioorganic & Medicinal Chemistry Letters, 2013, 23(10):3044-3050.
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