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Gestrinone

CAS No. 16320-04-0

Gestrinone ( R 2323 )

Catalog No. M20652 CAS No. 16320-04-0

Gestrinone is a synthetic androgen receptor agonist and ER and progesterone receptor antagonist used to treat endometriosis. It inhibits leiomyoma cells with an IC50 of 43.67 μM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 56 In Stock
10MG 90 In Stock
25MG 162 In Stock
50MG 243 In Stock
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Biological Information

  • Product Name
    Gestrinone
  • Note
    Research use only not for human use.
  • Brief Description
    Gestrinone is a synthetic androgen receptor agonist and ER and progesterone receptor antagonist used to treat endometriosis. It inhibits leiomyoma cells with an IC50 of 43.67 μM.
  • Description
    Gestrinone is a synthetic androgen receptor agonist and ER and progesterone receptor antagonist used to treat endometriosis. It inhibits leiomyoma cells with an IC50 of 43.67 μM.
  • Synonyms
    R 2323
  • Pathway
    Endocrinology/Hormones
  • Target
    Estrogen Receptor/ERR
  • Recptor
    ER
  • Research Area
    Others
  • Indication
    Endometriosis with or without accompanying sterility

Chemical Information

  • CAS Number
    16320-04-0
  • Formula Weight
    308.41
  • Molecular Formula
    C21H24O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:50 mg/mL (162.12 mM)
  • SMILES
    [H][C@@]12CC[C@@](O)(C#C)[C@@]1(CC)C=CC1=C3CCC(=O)C=C3CC[C@@]21[H]
  • Chemical Name
    (8S13S14S17S)-13-ethyl-17-ethynyl-17-hydroxy-126781314151617-decahydro-3H-cyclopenta[a]phenanthren-3-one

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Hui-Ling X Ning Y Jing W et al. Therapeutic effects of mifepristone combined withGestrinone on patients with endometriosis[J]. Pakistan Journal of Medical Sciences 2016 32(5).
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