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Home - Products - Endocrinology/Hormones - Estrogen Receptor/ERR - GSK-4716

GSK-4716

CAS No. 101574-65-6

GSK-4716 ( —— )

Catalog No. M20159 CAS No. 101574-65-6

GSK4716 is an ERRβ/γ agonist (IC50 = 2 μM) that can activate the receptor with similar potency as the protein ligand.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    GSK-4716
  • Note
    Research use only not for human use.
  • Brief Description
    GSK4716 is an ERRβ/γ agonist (IC50 = 2 μM) that can activate the receptor with similar potency as the protein ligand.
  • Description
    GSK4716 is an ERRβ/γ agonist (IC50 = 2 μM) that can activate the receptor with similar potency as the protein ligand.
  • Synonyms
    ——
  • Pathway
    Endocrinology/Hormones
  • Target
    Estrogen Receptor/ERR
  • Recptor
    ERRβ/γ
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    101574-65-6
  • Formula Weight
    282.34
  • Molecular Formula
    C17H18N2O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:100 mg/mL?(354.18 mM)
  • SMILES
    CC(C)c1ccc(cc1)\C=N\NC(=O)c1ccc(O)cc1
  • Chemical Name
    4-hydroxy-N-[(4-propan-2-ylphenyl)methylideneamino]benzamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Wang L Zuercher W J Consler T G et al. X-ray Crystal Structures of the Estrogen-related Receptor- Ligand Binding Domain in Three Functional States Reveal the Molecular Basis of Small Molecule Regulation[J]. Journal of Biological Chemistry 2006 281(49):37773-37781.
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