GSK-4716 ( —— )

Catalog No. M20159 CAS No. 101574-65-6

GSK4716 is an ERRβ/γ agonist (IC50 = 2 μM) that can activate the receptor with similar potency as the protein ligand.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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Biological Information

Product Name

GSK-4716
Note

Research use only not for human use.
Brief Description

GSK4716 is an ERRβ/γ agonist (IC50 = 2 μM) that can activate the receptor with similar potency as the protein ligand.
Description

GSK4716 is an ERRβ/γ agonist (IC50 = 2 μM) that can activate the receptor with similar potency as the protein ligand.
Synonyms

——
Pathway

Endocrinology/Hormones
Target

Estrogen Receptor/ERR
Recptor

ERRβ/γ
Research Area

——
Indication

——

Chemical Information

CAS Number

101574-65-6
Formula Weight

282.34
Molecular Formula

C17H18N2O2
Purity

>98% (HPLC)
Solubility

DMSO:100 mg/mL?(354.18 mM)
SMILES

CC(C)c1ccc(cc1)\C=N\NC(=O)c1ccc(O)cc1
Chemical Name

4-hydroxy-N-[(4-propan-2-ylphenyl)methylideneamino]benzamide

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Wang L Zuercher W J Consler T G et al. X-ray Crystal Structures of the Estrogen-related Receptor- Ligand Binding Domain in Three Functional States Reveal the Molecular Basis of Small Molecule Regulation[J]. Journal of Biological Chemistry 2006 281(49):37773-37781.

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