Cart
sales@molnova.com
Home - Products - Cell Cycle/DNA Damage - Topoisomerase - GW842166X

GW842166X

CAS No. 666260-75-9

GW842166X ( GW-842166X; 842166X; 842166 )

Catalog No. M18967 CAS No. 666260-75-9

GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM, shows no significant activity at CB1 receptor. Phase 2.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 39 In Stock
5MG 63 In Stock
10MG 113 In Stock
25MG 212 In Stock
50MG 313 In Stock
100MG 466 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
Group Booking Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    GW842166X
  • Note
    Research use only, not for human use.
  • Brief Description
    GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM, shows no significant activity at CB1 receptor. Phase 2.
  • Description
    GW 842166X is a cannabinoid receptor 2 (CB2) agonist potentially for the treatment of inflammatory pain.
  • Synonyms
    GW-842166X; 842166X; 842166
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    Topoisomerase
  • Recptor
    CB2
  • Research Area
    Others-Field
  • Indication
    ——

Chemical Information

  • CAS Number
    666260-75-9
  • Formula Weight
    449.25
  • Molecular Formula
    C18H17Cl2F3N4O2
  • Purity
    98%
  • Solubility
    DMSO : ≥ 83.3 mg/mL; 185.42 mM
  • SMILES
    FC(F)(F)C1=NC(NC2=CC=C(Cl)C=C2Cl)=NC=C1C(=O)NCC1CCOCC1
  • Chemical Name
    2-((2,4-dichlorophenyl)amino)-N-((tetrahydro-2H-pyran-4-yl)methyl)-4-(trifluoromethyl)pyrimidine-5-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Giblin GM, et al. J Med Chem, 2007, 50(11), 2597-2600.
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • ARN-21934

    ARN-21934 is a potent and selective inhibitor for human topoisomerase II α and topoisomerase II β. ARN-21934(IC50 = 2 μM) inhibits DNA relaxation as compared to the anticancer agent Etoposide (IC50=120 μM).

  • Ofloxacin

    Ofloxacin is a fluoroquinolone whose primary mechanism of action is inhibition of bacterial DNA gyrase.

  • Nalidixic acid sodiu...

    A synthetic 1,8-naphthyridine antimicrobial agent with a limited bacteriocidal spectrum.

Sign In Join Free