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GV150013
CAS No. 167355-22-8
GV150013( —— )
Catalog No. M34275 CAS No. 167355-22-8
GV150013 is an antagonist of cholecystokinin-2 (CCK2) receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 299 | Get Quote |
|
| 5MG | 455 | Get Quote |
|
| 10MG | 620 | Get Quote |
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| 25MG | 911 | Get Quote |
|
| 50MG | 1224 | Get Quote |
|
| 100MG | 1575 | Get Quote |
|
| 200MG | 2133 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameGV150013
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NoteResearch use only, not for human use.
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Brief DescriptionGV150013 is an antagonist of cholecystokinin-2 (CCK2) receptor.
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DescriptionGV-150013 is a selective CCK-B receptor antagonist. GV-150013 has sleep aid effect.
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In Vitro——
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In VivoAnimal Model:Old rats .Dosage:0.5 μg/kg, 5μg/kg, 60μg/kg Administration:Intraperitoneal injection, Once Result:The duration of REM sleep and non-REM sleep was longer than that of control.
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Synonyms——
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PathwayGPCR/G Protein
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TargetCholecystokinin Receptor
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Recptorcholecystokinin
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Research Area——
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Indication——
Chemical Information
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CAS Number167355-22-8
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Formula Weight534.65
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Molecular FormulaC33H34N4O3
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Purity>98% (HPLC)
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Solubility——
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SMILESC(C12CC3CC(C1)CC(C2)C3)N4C=5C(N(C(=O)[C@H](NC(NC6=CC=CC=C6)=O)C4=O)C7=CC=CC=C7)=CC=CC5
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Crespi F. Cholecystokinin-B (CCK-B) receptor antagonists improve "aged" sleep: a new class of sleep modulators? Methods Find Exp Clin Pharmacol. 1999 Jan-Feb;21(1):31-8.?
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