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GSK5182
CAS No. 877387-37-6
GSK5182 ( —— )
Catalog No. M21654 CAS No. 877387-37-6
GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)?.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 61 | In Stock |
|
| 5MG | 87 | In Stock |
|
| 10MG | 140 | In Stock |
|
| 25MG | 260 | In Stock |
|
| 50MG | 394 | In Stock |
|
| 100MG | 582 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameGSK5182
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NoteResearch use only not for human use.
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Brief DescriptionGSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)?.
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DescriptionGSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)?.
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetEstrogen Receptor/ERR
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RecptorERRγ
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Research Area——
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Indication——
Chemical Information
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CAS Number877387-37-6
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Formula Weight417.55
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Molecular FormulaC27H31NO3
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Purity>98% (HPLC)
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Solubility——
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SMILESCN(C)CCOc1ccc(cc1)C(\c1ccc(O)cc1)=C(\CCCO)c1ccccc1
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Chemical Name4-[(Z)-1-[4-(2-dimethylaminoethoxy)phenyl]-5-hydroxy-2-phenylpent-1-enyl]phenol
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Kim JH et al. Estrogen-related receptor γ is upregulated in liver cancer and its inhibition suppresses livercancer cell proliferation via induction of p21 and p27. Exp Mol Med. 2016 Mar 4;48:e213.
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