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GSK2656157
CAS No. 1337532-29-2
GSK2656157 ( GSK2656157; GSK 2656157; GSK-2656157 )
Catalog No. M11351 CAS No. 1337532-29-2
GSK2656157 is an ATP-competitive and highly selective inhibitor of PERK with IC50 of 0.9 nM in a cell-free assay.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 29 | In Stock |
|
| 5MG | 46 | In Stock |
|
| 10MG | 67 | In Stock |
|
| 25MG | 131 | In Stock |
|
| 50MG | 245 | In Stock |
|
| 100MG | 443 | In Stock |
|
| 200MG | 599 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameGSK2656157
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NoteResearch use only, not for human use.
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Brief DescriptionGSK2656157 is an ATP-competitive and highly selective inhibitor of PERK with IC50 of 0.9 nM in a cell-free assay.
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DescriptionGSK2656157 is an ATP-competitive and highly selective inhibitor of PERK with IC50 of 0.9 nM in a cell-free assay, 500-fold greater against a panel of 300 kinases.
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SynonymsGSK2656157; GSK 2656157; GSK-2656157
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PathwayMAPK/ERK Signaling
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TargetERK
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RecptorPERK
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1337532-29-2
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Formula Weight416.45
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Molecular FormulaC23H21FN6O
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Purity>98%(HPLC)
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SolubilityDMSO: 32 mg/mL (76.83 mM)
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SMILESCC1=CC=CC(CC(N2CCC3=C2C=CC(C4=CN(C)C5=NC=NC(N)=C54)=C3F)=O)=N1
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Chemical Name1-(5-(4-amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)-4-fluoroindolin-1-yl)-2-(6-methylpyridin-2-yl)ethanone
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Atkins C, et al. Y Res, 2013, 73(6), 1993-2002.
molnova catalog
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