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GSK2193874
CAS No. 1336960-13-4
GSK2193874 ( —— )
Catalog No. M20323 CAS No. 1336960-13-4
GSK2193874 was identified as a selective orally active TRPV4 blocker.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 47 | In Stock |
|
| 5MG | 67 | In Stock |
|
| 10MG | 116 | In Stock |
|
| 25MG | 233 | In Stock |
|
| 50MG | 383 | In Stock |
|
| 100MG | 570 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameGSK2193874
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NoteResearch use only not for human use.
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Brief DescriptionGSK2193874 was identified as a selective orally active TRPV4 blocker.
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DescriptionGSK2193874 was identified as a selective orally active TRPV4 blocker.
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetTRP/TRPV Channel
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RecptorTRPV4
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Research Area——
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Indication——
Chemical Information
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CAS Number1336960-13-4
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Formula Weight691.6
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Molecular FormulaC37H38BrF3N4O
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Purity>98% (HPLC)
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SolubilityDMSO:100 mg/mL?(144.59 mM)
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SMILESFC(F)(F)c1cccc(c1)-c1nc2cc(Br)ccc2c(C(=O)NC2(CC2)c2ccccc2)c1CN1CCC(CC1)N1CCCCC1
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Chemical Name7-bromo-N-(1-phenylcyclopropyl)-3-[(4-piperidin-1-ylpiperidin-1-yl) methyl]-2-[3-(trifluoromethyl)phenyl]quinoline-4-carboxamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Cheung M Bao W Behm D J et al. Discovery of GSK2193874: An Orally Active Potent and Selective Blocker of Transient Receptor Potential Vanilloid 4[J]. ACS Medicinal Chemistry Letters 2017:acsmedchemlett.7b00094.
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