GSK2193874 ( —— )

Catalog No. M20323 CAS No. 1336960-13-4

GSK2193874 was identified as a selective orally active TRPV4 blocker.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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5MG	67	In Stock
10MG	116	In Stock
25MG	233	In Stock
50MG	383	In Stock
100MG	570	In Stock
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Biological Information

Product Name

GSK2193874
Note

Research use only not for human use.
Brief Description

GSK2193874 was identified as a selective orally active TRPV4 blocker.
Description

GSK2193874 was identified as a selective orally active TRPV4 blocker.
Synonyms

——
Pathway

Membrane Transporter/Ion Channel
Target

TRP/TRPV Channel
Recptor

TRPV4
Research Area

——
Indication

——

Chemical Information

CAS Number

1336960-13-4
Formula Weight

691.6
Molecular Formula

C37H38BrF3N4O
Purity

>98% (HPLC)
Solubility

DMSO:100 mg/mL?(144.59 mM)
SMILES

FC(F)(F)c1cccc(c1)-c1nc2cc(Br)ccc2c(C(=O)NC2(CC2)c2ccccc2)c1CN1CCC(CC1)N1CCCCC1
Chemical Name

7-bromo-N-(1-phenylcyclopropyl)-3-[(4-piperidin-1-ylpiperidin-1-yl) methyl]-2-[3-(trifluoromethyl)phenyl]quinoline-4-carboxamide

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Cheung M Bao W Behm D J et al. Discovery of GSK2193874: An Orally Active Potent and Selective Blocker of Transient Receptor Potential Vanilloid 4[J]. ACS Medicinal Chemistry Letters 2017:acsmedchemlett.7b00094.

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