GSK-812

CAS No. 630407-66-8

GSK-812 ( GSK812 )

Catalog No. M15383 CAS No. 630407-66-8

GSK-812 is a potent neuroprotectant that can induce GDNF in normal and diseased retina.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    GSK-812
  • Note
    Research use only, not for human use.
  • Brief Description
    GSK-812 is a potent neuroprotectant that can induce GDNF in normal and diseased retina.
  • Description
    GSK-812 is a potent neuroprotectant that can induce GDNF in normal and diseased retina, shows has polypharmacology antagonizing multiple receptors, including D2 and D3 receptors, and 5-HT2A, 2C, and 5-HT6 receptors.
  • Synonyms
    GSK812
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    630407-66-8
  • Formula Weight
    472.00
  • Molecular Formula
    C25H26ClNO4S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CN1CCC2=CC(=C(C=C2CC1)S(=O)(=O)C3=CC=C(C=C3)OCC4=CC=C(C=C4)Cl)OC
  • Chemical Name
    7-[4-(4-chloro-benzyloxy)-benzenesulfonyl]-8-methoxy-3-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Baranov P, et al. J Ocul Pharmacol Ther. 2017 Jun;33(5):412-422.
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