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GSK-812
CAS No. 630407-66-8
GSK-812( GSK812 )
Catalog No. M15383 CAS No. 630407-66-8
GSK-812 is a potent neuroprotectant that can induce GDNF in normal and diseased retina.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameGSK-812
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NoteResearch use only, not for human use.
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Brief DescriptionGSK-812 is a potent neuroprotectant that can induce GDNF in normal and diseased retina.
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DescriptionGSK-812 is a potent neuroprotectant that can induce GDNF in normal and diseased retina, shows has polypharmacology antagonizing multiple receptors, including D2 and D3 receptors, and 5-HT2A, 2C, and 5-HT6 receptors.
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In Vitro——
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In Vivo——
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SynonymsGSK812
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor5-HT Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number630407-66-8
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Formula Weight471.996
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Molecular FormulaC25H26ClNO4S
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Purity>98% (HPLC)
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Solubility——
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SMILESCN1CCC2=CC(=C(C=C2CC1)S(=O)(=O)C3=CC=C(C=C3)OCC4=CC=C(C=C4)Cl)OC
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Chemical Name7-[4-(4-chloro-benzyloxy)-benzenesulfonyl]-8-methoxy-3-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Baranov P, et al. J Ocul Pharmacol Ther. 2017 Jun;33(5):412-422.
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