GS967

CAS No. 1262618-39-2

GS967( GS967 | GS-967 | GS 967 | GS458967 )

Catalog No. M11095 CAS No. 1262618-39-2

GS967 is a novel, potent, and selective inhibitor of cardiac late sodium current(late INa).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 27 In Stock
5MG 43 In Stock
10MG 65 In Stock
25MG 146 In Stock
50MG 268 In Stock
100MG 470 In Stock
200MG 680 In Stock
500MG 1053 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    GS967
  • Note
    Research use only, not for human use.
  • Brief Description
    GS967 is a novel, potent, and selective inhibitor of cardiac late sodium current(late INa).
  • Description
    GS967 is a novel, potent, and selective inhibitor of cardiac late sodium current(late INa); inhibits ATX-II-induced late I(Na) in ventricular myocytes and isolated hearts with IC(50) values of 0.13 and 0.21 μM, respectively.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    GS967 | GS-967 | GS 967 | GS458967
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    Sodium Channel
  • Recptor
    late?INa?,isolated hearts| late?INa?,ventricular myocytes
  • Research Area
    Cardiovascular Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    1262618-39-2
  • Formula Weight
    347.22
  • Molecular Formula
    C14H7F6N3O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 10 mM
  • SMILES
    FC(C1=NN=C2C=CC(C3=CC=C(OC(F)(F)F)C=C3)=CN21)(F)F
  • Chemical Name
    6-(4-(trifluoromethoxy)phenyl)-3-(trifluoromethyl)(1,2,4)triazolo(4,3-a)pyridine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Belardinelli L, et al. J Pharmacol Exp Ther. 2013 Jan;344(1):23-32.
molnova catalog
related products
  • Phenazopyridine hydr...

    Phenazopyridine hydrochloride is a local analgesic that has been used in urinary tract disorders.

  • Levobupivacaine

    Levobupivacaine is an amino-amide local anaesthetic drug belonging to the family of n-alkylsubstituted pipecoloxylidide.

  • λ-Cyhalothrin

    lambda-Cyhalothrin is a high efficiency, broad-spectrum type II synthetic pyrethroid insecticide containing α-cyano group.lambda-Cyhalothrin is used to control a wide range of pests in a variety of applications.lambda-Cyhalothrin is a neurotoxin that targets sodium channels in the membranes of neurons in the central nervous system.