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FTIDC
CAS No. 873551-53-2
FTIDC ( FTIDC )
Catalog No. M17636 CAS No. 873551-53-2
FTIDC is a highly potent and selective allosteric antagonist of mGluR1 receptors and shows very weak potency against human and rat mGluR5 receptors.
Purity : 95%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 140 | In Stock |
|
| 5MG | 215 | In Stock |
|
| 10MG | 340 | In Stock |
|
| 25MG | 565 | In Stock |
|
| 50MG | 797 | In Stock |
|
| 100MG | 1071 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameFTIDC
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NoteResearch use only, not for human use.
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Brief DescriptionFTIDC is a highly potent and selective allosteric antagonist of mGluR1 receptors and shows very weak potency against human and rat mGluR5 receptors.
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DescriptionFTIDC is a highly potent and selective allosteric antagonist of mGluR1 receptors and shows very weak potency against human and rat mGluR5 receptors. The inhibition of FTIDC for mGluR1 receptors is shown to be in noncompetitive manner and displays IC50 values of 5.8 and 3.1 nM for human and mouse mGluR1 expressed in CHO cells respectively.
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SynonymsFTIDC
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PathwayOthers
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TargetOther Targets
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RecptormGluR1
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Research Area——
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Indication——
Chemical Information
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CAS Number873551-53-2
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Formula Weight358.42
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Molecular FormulaC18H23FN6O
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Purity95%
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Solubility——
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SMILESC1CC(=CCN1C(=O)N(C(C)C)C)c1nnn(c1C)c1c(nccc1)F
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Chemical Name4-[1-(2-Fluoropyridin-3-yl)-5-methyl-1H-1,2,3-triazol-4-yl]-N-isopropyl-N-methyl-3,6-dihydropyridine-1(2H)-carboxamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Ito S, et al. Bioorg Med Chem. 2008 Nov 15;16(22):9817-29.
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