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FAK-IN-10
CAS No. 491839-65-7
FAK-IN-10( —— )
Catalog No. M37079 CAS No. 491839-65-7
FAK-IN-10 is an inhibitor of FAK (IC50: 76.3 μM) and demonstrates antitumor activity in MCF-7 and A431 cell lines with IC50 values of 4.23 μM and 0.78 μM, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 88 | Get Quote |
|
| 5MG | 132 | Get Quote |
|
| 10MG | 211 | Get Quote |
|
| 25MG | 348 | Get Quote |
|
| 50MG | 490 | Get Quote |
|
| 100MG | 682 | Get Quote |
|
| 500MG | 1377 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameFAK-IN-10
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NoteResearch use only, not for human use.
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Brief DescriptionFAK-IN-10 is an inhibitor of FAK (IC50: 76.3 μM) and demonstrates antitumor activity in MCF-7 and A431 cell lines with IC50 values of 4.23 μM and 0.78 μM, respectively.
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DescriptionFAK-IN-10 is an inhibitor of FAK with an IC50 of 76.3 μM. FAK-IN-10 exhibits antitumor activity against MCF-7 and A431 cell lines with IC50s of 4.23 and 0.78 μM,respectively.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetFAK
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RecptorFAK
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Research Area——
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Indication——
Chemical Information
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CAS Number491839-65-7
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Formula Weight376.23
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Molecular FormulaC15H10BrN3O2S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 20 mg/mL (53.16 mM; Ultrasonic (<60°C)
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SMILESO=C(C1=CC=C(Br)C=C1)CSC2=NN=C(O2)C=3C=CN=CC3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Zhang LR, et al. Synthesis, biological evaluation and molecular docking studies of novel 2-(1,3,4-oxadiazol-2-ylthio)-1-phenylethanone derivatives. Bioorg Med Chem. 2012 Jun 1;20(11):3615-21.?
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FAK-IN-10
FAK-IN-10 is an inhibitor of FAK (IC50: 76.3 μM) and demonstrates antitumor activity in MCF-7 and A431 cell lines with IC50 values of 4.23 μM and 0.78 μM, respectively.
