Erastin2

CAS No. 1695533-44-8

Erastin2( —— )

Catalog No. M34807 CAS No. 1695533-44-8

Erastin2 is a ferroptosis inducer and inhibitor of the system xc- cystine/glutamate transporter.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 102 Get Quote
5MG 155 Get Quote
10MG 250 Get Quote
25MG 410 Get Quote
50MG 655 Get Quote
100MG 981 Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    Erastin2
  • Note
    Research use only, not for human use.
  • Brief Description
    Erastin2 is a ferroptosis inducer and inhibitor of the system xc- cystine/glutamate transporter.
  • Description
    Erastin2 is a ferroptosis inducer and a potent, selective inhibitor of the system xc(-) cystine/glutamate transporter.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Apoptosis
  • Target
    Ferroptosis
  • Recptor
    Ferroptosis
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1695533-44-8
  • Formula Weight
    623.14
  • Molecular Formula
    C36H35ClN4O4
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (160.48 mM; Ultrasonic )
  • SMILES
    CC(C)Oc1ccc(cc1-n1c(CN2CCN(CC2)C(=O)COc2ccc(Cl)cc2)nc2ccccc2c1=O)-c1ccccc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Cao JY, et al. A Genome-wide Haploid Genetic Screen Identifies Regulators of Glutathione Abundance and Ferroptosis Sensitivity. Cell Rep. 2019 Feb 5;26(6):1544-1556.e8. ?
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