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Ensitrelvir
CAS No. 2647530-73-0
Ensitrelvir( S-217622 )
Catalog No. M28855 CAS No. 2647530-73-0
Ensitrelvir.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 10MG | 45 | In Stock |
|
| 25MG | 104 | In Stock |
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| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
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Biological Information
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Product NameEnsitrelvir
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NoteResearch use only, not for human use.
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Brief DescriptionEnsitrelvir.
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DescriptionEnsitrelvir.(In Vitro):The EC50 values for SARS-CoV and MERS-CoV were 0.21 and 1.4 μM respectively. In a cytopathic effect (cpe)-inhibition assay of SARS-CoV-2 infected VeroE6/TMPRSS2 cells, Ensitrelvir shows the EC50 values are approximately 0.4 μM for both wild-type virus and Alpha, Beta, Gamma and Delta variants.(In Vivo):Ensitrelvir inhibits intrapulmonary replication of SARS-CoV-2 in mice in a dose-dependent manner.
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In Vitro——
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In Vivo——
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SynonymsS-217622
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PathwayOthers
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TargetOther Targets
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RecptorCOX-2|5-Lipoxygenase
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Research Area——
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Indication——
Chemical Information
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CAS Number2647530-73-0
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Formula Weight531.88
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Molecular FormulaC22H17ClF3N9O2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 50 mg/mL (94.01 mM)
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SMILESCn1nc(cc(c(/N=C(\NC(N2Cc3nn(C)cn3)=O)/N(Cc(cc(c(F)c3)F)c3F)C2=O)c2)Cl)c2c1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Kirchner T, et al. Evaluation of the antiinflammatory activity of a dual cyclooxygenase-2 selective/5-lipoxygenase inhibitor, RWJ 63556, in a canine model of inflammation. J Pharmacol Exp Ther. 1997 Aug;282(2):1094-101.
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