
Endoxifen
CAS No. 112093-28-4
Endoxifen( —— )
Catalog No. M10432 CAS No. 112093-28-4
A metabolite of tamoxifen, orally active non-steroidal selective estrogen receptor modulator (SERM) for the treatment of estrogen receptor-positive breast cancer.
Purity : >98% (HPLC)






Size | Price / USD | Stock | Quantity |
2MG | 73 | In Stock |
![]() ![]() |
5MG | 120 | In Stock |
![]() ![]() |
10MG | 192 | In Stock |
![]() ![]() |
25MG | 356 | In Stock |
![]() ![]() |
50MG | 555 | In Stock |
![]() ![]() |
100MG | Get Quote | In Stock |
![]() ![]() |
200MG | Get Quote | In Stock |
![]() ![]() |
500MG | Get Quote | In Stock |
![]() ![]() |
1G | Get Quote | In Stock |
![]() ![]() |
Biological Information
-
Product NameEndoxifen
-
NoteResearch use only, not for human use.
-
Brief DescriptionA metabolite of tamoxifen, orally active non-steroidal selective estrogen receptor modulator (SERM) for the treatment of estrogen receptor-positive breast cancer.
-
DescriptionA metabolite of tamoxifen, orally active non-steroidal selective estrogen receptor modulator (SERM) for the treatment of estrogen receptor-positive breast cancer.Breast Cancer Phase 1 Clinical.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayEndocrinology/Hormones
-
TargetEstrogen Receptor/ERR
-
RecptorER|ERR|hERGPotassiumChannel
-
Research AreaCancer
-
IndicationBreast Cancer
Chemical Information
-
CAS Number112093-28-4
-
Formula Weight373.4874
-
Molecular FormulaC25H27NO2
-
Purity>98% (HPLC)
-
Solubility10 mM in DMSO
-
SMILESCCC(=C(C1=CC=C(C=C1)O)C2=CC=C(C=C2)OCCNC)C3=CC=CC=C3
-
Chemical NamePhenol, 4-[(1Z)-1-[4-[2-(methylamino)ethoxy]phenyl]-2-phenyl-1-buten-1-yl]-
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Brauch H, et al. Clin Chem. 2009 Oct;55(10):1770-82.
2. Markopoulos C, et al. World J Clin Oncol. 2014 Aug 10;5(3):374-81.
3. Mugundu GM, et al. Drug Metab Dispos. 2012 Feb;40(2):389-96.
molnova catalog



related products
-
PHTPP
A potent, selective antagonist of estrogen ERβ receptor; exhibits 36-fold selective for ERβ, and is fully effective as an ERα antagonist.
-
Ethynodiol diacetate
Ethynodiol diacetate is one of the first synthetic progestogens used in contraceptive pills.
-
Hydroxyprogesterone
17-Hydroxyprogesterone (17-OHP) is an endogenous progestogen as well as chemical intermediate in the biosynthesis of other steroid hormones.