Desmethyl-VS-5584

CAS No. 1246535-95-4

Desmethyl-VS-5584( Desmethyl-VS-5584 | Desmethyl-VS5584 )

Catalog No. M17217 CAS No. 1246535-95-4

Desmethyl-VS-5584 is a dimethyl analog of VS-5584, which is a novel and highly selective PI3K/mTOR kinase inhibitor for the treatment of cancer.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 91 In Stock
5MG 145 In Stock
10MG 257 In Stock
25MG 430 In Stock
50MG 621 In Stock
100MG 883 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Desmethyl-VS-5584
  • Note
    Research use only, not for human use.
  • Brief Description
    Desmethyl-VS-5584 is a dimethyl analog of VS-5584, which is a novel and highly selective PI3K/mTOR kinase inhibitor for the treatment of cancer.
  • Description
    Desmethyl-VS-5584 is a demethyl analogue of VS-5584, which is a novel and highly selective PI3K/mTOR kinase inhibitor for the treatment of cancer.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Desmethyl-VS-5584 | Desmethyl-VS5584
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    PARP
  • Recptor
    mTOR| PI3K
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1246535-95-4
  • Formula Weight
    340.39
  • Molecular Formula
    C16H20N8O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Nc1ncc(c2c3ncn(C(C)C)c3nc(N3CCOCC3)n2)cn1
  • Chemical Name
    5-[9-(1-Methylethyl)-2-(4-morpholinyl)-9H-purin-6-yl]-2-pyrimidinamine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Shao Z,et al. VS-5584, a Novel PI3K-mTOR Dual Inhibitor, Inhibits Melanoma Cell Growth In Vitro and In Vivo. PLoS One. 2015 Jul 23;10(7).
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