Delpazolid
CAS No. 1219707-39-7
Delpazolid ( LCB01-0371;LCB 01-0371 )
Catalog No. M10827 CAS No. 1219707-39-7
A novel oxazolidinone antibiotic that shows good antibacterial activity (MSSA MIC50=1 ug/mL).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 72 | In Stock |
|
10MG | 125 | In Stock |
|
25MG | 260 | In Stock |
|
50MG | 447 | In Stock |
|
100MG | 624 | In Stock |
|
500MG | 1305 | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
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Product NameDelpazolid
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NoteResearch use only, not for human use.
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Brief DescriptionA novel oxazolidinone antibiotic that shows good antibacterial activity (MSSA MIC50=1 ug/mL).
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DescriptionA novel oxazolidinone antibiotic that shows good antibacterial activity (MSSA MIC50=1 ug/mL); potently inhibits MSSA and MRSA clinical isolates with MIC of 0.5-2 and 0.5-4 ug/mL, respectively; shows more-potent protective effects (MSSA ED50=4.53 mg/kg) than Linezolid against systemic infections caused by Gram-positive and Gram-negative bacteria in mice model.Bacterial Infection Preclinical
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SynonymsLCB01-0371;LCB 01-0371
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PathwayGPCR/G Protein
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TargetAntibacterial
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RecptorOthers
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Research AreaInfection
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IndicationBacterial Infection
Chemical Information
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CAS Number1219707-39-7
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Formula Weight308.31
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Molecular FormulaC14H17FN4O3
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESO=C1O[C@@H](CO)CN1C2=CC=C(N3C=NN(C)CC3)C(F)=C2
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Chemical Name(5R)-3-[3-fluoro-4-(1-methyl-5,6-dihydro-1,2,4-triazin-4(1H)-yl)phenyl]-5-(hydroxymethyl)-1,3-oxazolidin-2-one
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Jeong JW, et al. Antimicrob Agents Chemother. 2010 Dec;54(12):5359-62.
2. Kim TS, et al. Antimicrob Agents Chemother. 2017 Aug 24;61(9). pii: e02752-16.
3. Choi Y, et al. J Antimicrob Chemother. 2017 Oct 23. doi: 10.1093/jac/dkx367.
2. Kim TS, et al. Antimicrob Agents Chemother. 2017 Aug 24;61(9). pii: e02752-16.
3. Choi Y, et al. J Antimicrob Chemother. 2017 Oct 23. doi: 10.1093/jac/dkx367.
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