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Delamanid
CAS No. 681492-22-8
Delamanid( OPC67683 | OPC-67683 | OPC 67683 )
Catalog No. M15601 CAS No. 681492-22-8
A mycolic acid biosynthesis inhibitor found to be free of mutagenicity and to possess highly potent activity against tuberculosis.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 35 | In Stock |
|
| 10MG | 58 | In Stock |
|
| 25MG | 113 | In Stock |
|
| 50MG | 203 | In Stock |
|
| 100MG | 329 | In Stock |
|
| 500MG | 770 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameDelamanid
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NoteResearch use only, not for human use.
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Brief DescriptionA mycolic acid biosynthesis inhibitor found to be free of mutagenicity and to possess highly potent activity against tuberculosis.
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DescriptionA mycolic acid biosynthesis inhibitor found to be free of mutagenicity and to possess highly potent activity against tuberculosis, including MDR-TB; shows MIC of 0.006-0.024 ug/mL in vitro and highly effective therapeutic activity at low doses in vivo.
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In Vitro——
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In Vivo——
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SynonymsOPC67683 | OPC-67683 | OPC 67683
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PathwayGPCR/G Protein
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TargetAntibacterial
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RecptorAntifection
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Research AreaInfection
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Indication——
Chemical Information
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CAS Number681492-22-8
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Formula Weight534.4844
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Molecular FormulaC25H25F3N4O6
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 30 mg/mL
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SMILESFC(F)(F)OC1=CC=C(OC2CCN(C3=CC=C(OC[C@@]4(C)CN5C(O4)=NC([N+]([O-])=O)=C5)C=C3)CC2)C=C1
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Chemical NameImidazo[2,1-b]oxazole, 2,3-dihydro-2-methyl-6-nitro-2-[[4-[4-[4-(trifluoromethoxy)phenoxy]-1-piperidinyl]phenoxy]methyl]-, (2R)-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Matsumoto M, et al. PLoS Med. 2006 Nov;3(11):e466.
2. Li X, et al. Bioorg Med Chem Lett. 2008 Apr 1;18(7):2256-62.
3. Hurdle JG, et al. J Antimicrob Chemother. 2008 Nov;62(5):1037-45.
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