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DS08210767
CAS No. 2376334-75-5
DS08210767( —— )
Catalog No. M32894 CAS No. 2376334-75-5
DS08210767 is a highly potent, orally bioavailable PTHR1 antagonist with an IC50 of 90 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 196 | Get Quote |
|
| 5MG | 306 | Get Quote |
|
| 10MG | 443 | Get Quote |
|
| 25MG | 638 | Get Quote |
|
| 50MG | 878 | Get Quote |
|
| 100MG | 1170 | Get Quote |
|
| 500MG | 2349 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameDS08210767
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NoteResearch use only, not for human use.
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Brief DescriptionDS08210767 is a highly potent, orally bioavailable PTHR1 antagonist with an IC50 of 90 nM.
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DescriptionDS08210767 is a highly potent, orally bioavailable PTHR1 antagonist with IC50 of 90 nM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetTHR
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RecptorThyroid hormone receptor(THR)
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Research Area——
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Indication——
Chemical Information
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CAS Number2376334-75-5
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Formula Weight513.67
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Molecular FormulaC31H39N5O2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 5 mg/mL (9.73 mM; Ultrasonic (<80°C)
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SMILESCC1(C)N=C(C2CCCCC2)c2ccc(cc2N(c2ccc(NCCNC3CCOCC3)cc2)C1=O)C#N
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Arai Y, et al. Discovery of novel PTHR1 antagonists: Design, synthesis, and structure activity relationships. Bioorg Med Chem Lett. 2019 Sep 15;29(18):2613-2616.?
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