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DRAK2-IN-16
CAS No. 871837-60-4
DRAK2-IN-16( —— )
Catalog No. M16339 CAS No. 871837-60-4
DRAK2-IN-116 is a potent, selective DRAK2 inhibitor with IC50 of 3 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 194 | Get Quote |
|
| 50MG | 896 | Get Quote |
|
| 100MG | 1566 | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameDRAK2-IN-16
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NoteResearch use only, not for human use.
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Brief DescriptionDRAK2-IN-116 is a potent, selective DRAK2 inhibitor with IC50 of 3 nM.
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DescriptionDRAK2-IN-116 is a potent, selective DRAK2 inhibitor with IC50 of 3 nM, shows weak inhibition for DRAK1 (IC50=51 nM) and no significant activity against DAPK1/2/3 (IC50>1 uM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayApoptosis
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TargetDAPK
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RecptorDAPK
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Research Area——
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Indication——
Chemical Information
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CAS Number871837-60-4
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Formula Weight376.416
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Molecular FormulaC21H20N4O3
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (265.67 mM)
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SMILESCCCCC(NC1=CC2=C(NC(/C2=C3NC4=C(C=CC=C4)C\3=N\O)=O)C=C1)=O
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Chemical NameN-((2Z,3E)-3-(hydroxyimino)-2'-oxo-[2,3'-biindolinylidene]-5'-yl)pentanamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Jung ME, et al. Bioorg Med Chem Lett. 2016 Jun 1;26(11):2719-23.
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