Cart
sales@molnova.com
Home - Products - Endocrinology/Hormones - 5-HT Receptor - Cerlapirdine

Cerlapirdine

CAS No. 925448-93-7

Cerlapirdine( SAM531 | SAM-531 | SAM 531 | PF-05212365 | P -05212365 | WAY-262,531 )

Catalog No. M27966 CAS No. 925448-93-7

Cerlapirdine is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine is already in clinical development for the treatment of cognitive disorders related to Alzheimer's disease and schizophrenia. It works by acting as a selective 5-HT6 receptor antagonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 160 Get Quote
10MG 260 Get Quote
25MG 515 Get Quote
50MG 740 Get Quote
100MG 1017 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote
Group Booking Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    Cerlapirdine
  • Note
    Research use only, not for human use.
  • Brief Description
    Cerlapirdine is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine is already in clinical development for the treatment of cognitive disorders related to Alzheimer's disease and schizophrenia. It works by acting as a selective 5-HT6 receptor antagonist.
  • Description
    Cerlapirdine is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine is already in clinical development for the treatment of cognitive disorders related to Alzheimer's disease and schizophrenia. It works by acting as a selective 5-HT6 receptor antagonist.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    SAM531 | SAM-531 | SAM 531 | PF-05212365 | P -05212365 | WAY-262,531
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    hSmo|mSmo
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    925448-93-7
  • Formula Weight
    409.5
  • Molecular Formula
    C22H23N3O3S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 41.67 mg/mL (101.76 mM)
  • SMILES
    CN(C)CCCOc1ccc2n[nH]c(c2c1)S(=O)(=O)c1cccc2ccccc12
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Lauressergues E, et al. Pharmacological evaluation of a series of smoothened antagonists in signaling pathways and after topical application in a depilated mouse model. Pharmacol Res Perspect. 2016 Mar 4;4(2):e00214.
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • Sarpogrelate hydroch...

    A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A; also shows binding affinity for 5-HT2B.

  • R-Lorcaserin hydroch...

    R-Lorcaserin hydrochloride hemihydrate is a selective 5HT2C serotonin receptor agonist.

  • Lurasidone

    Lurasidone is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6.75 nM).

Sign In Join Free