Carebastine
CAS No. 90729-42-3
Carebastine ( —— )
Catalog No. M26088 CAS No. 90729-42-3
Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 33 | In Stock |
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5MG | 53 | In Stock |
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10MG | 87 | In Stock |
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25MG | 177 | In Stock |
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50MG | 264 | In Stock |
|
100MG | 393 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
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Biological Information
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Product NameCarebastine
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NoteResearch use only, not for human use.
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Brief DescriptionCarebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.
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DescriptionCarebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.(In Vitro):Carebastine inhibits VEGF-induced HPAEC and HUVEC proliferation, migration, and angiogenesis in a dose-dependent manner . Carebastine suppresses the expression of macrophage migration inhibitory factor .
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Synonyms——
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PathwayGPCR/G Protein
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TargetHistamine Receptor
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RecptorParasite
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Research Area——
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Indication——
Chemical Information
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CAS Number90729-42-3
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Formula Weight499.7
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Molecular FormulaC32H37NO4
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Purity>98% (HPLC)
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Solubility——
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SMILESCC(C)(C(O)=O)c1ccc(cc1)C(=O)CCCN1CCC(CC1)OC(c1ccccc1)c1ccccc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Computer-aided analysis of phytochemicals as potential dengue virus inhibitors based on molecular docking, ADMET and DFT studies.J Vector Borne Dis. 2017 Jul-Sep;54(3):255-262.
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