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CaSR-IN-10a

CAS No. 478963-79-0

CaSR-IN-10a( —— )

Catalog No. M14596 CAS No. 478963-79-0

A potent CaSR antagonist with IC50 of 4.4 nM in CaSR FLIPR assay.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    CaSR-IN-10a
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent CaSR antagonist with IC50 of 4.4 nM in CaSR FLIPR assay.
  • Description
    A potent CaSR antagonist with IC50 of 4.4 nM in CaSR FLIPR assay.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    CaSR
  • Recptor
    CaSR
  • Research Area
    Other Indications
  • Indication
    ——

Chemical Information

  • CAS Number
    478963-79-0
  • Formula Weight
    360.4489
  • Molecular Formula
    C23H24N2O2
  • Purity
    >98% (HPLC)
  • Solubility
    10 mM in DMSO
  • SMILES
    CC(C)C1=CC=C(C=C1)C2=NC(=O)N(C3=C2C=C(C=C3)OCC#C)C(C)C
  • Chemical Name
    2(1H)-Quinazolinone, 1-(1-methylethyl)-4-[4-(1-methylethyl)phenyl]-6-(2-propyn-1-yloxy)-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Widler L, et al. J Med Chem. 2010 Mar 11;53(5):2250-63.
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