CZEN-002

CAS No. 581-05-5

CZEN-002 ( α-Melanocyte-Stimulating Hormone (MSH) amide )

Catalog No. M21154 CAS No. 581-05-5

CZEN-002 is amide stimulates melanocortin 1 receptor that results in the activation of adenylyl cyclase.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 146 In Stock
10MG 255 In Stock
25MG 430 In Stock
50MG 618 In Stock
100MG 897 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    CZEN-002
  • Note
    Research use only not for human use.
  • Brief Description
    CZEN-002 is amide stimulates melanocortin 1 receptor that results in the activation of adenylyl cyclase.
  • Description
    CZEN-002 is amide stimulates melanocortin 1 receptor that results in the activation of adenylyl cyclase.
  • Synonyms
    α-Melanocyte-Stimulating Hormone (MSH) amide
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    Adenylate Cyclase
  • Recptor
    Adenylyl cyclase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    581-05-5
  • Formula Weight
    1664.88
  • Molecular Formula
    C77H109N21O19S
  • Purity
    >98% (HPLC)
  • Solubility
    H2O:50 mg/mL (30.03 mM; Need ultrasonic)
  • SMILES
    OC[C@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CO)NC(C)=O)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](Cc2cncn2)C(=O)N[C@@H](Cc3ccccc3)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc5cnc4ccccc45)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N6CCC[C@H]6C(=O)N[C@H](C(N)=O)C(C)C
  • Chemical Name
    (4S7S10S13S16S22S)-7-((1H-imidazol-4-yl)methyl)-16-((1H-indol-3-yl)methyl)-26-amino-22-((S)-2-(((S)-1-amino-3-methyl-1-oxobutan-2-yl)carbamoyl)pyrrolidine-1-carbonyl)-10-benzyl-13-(3-guanidinopropyl)-4-((2S5S8S11S)-8-(4-hydroxybenzyl)-511-bis(hydroxymethyl)-2-(2-(methylthio)ethyl)-471013-tetraoxo-36912-tetraazatetradecanamido)-5811141720-hexaoxo-6912151821-hexaazahexacosanoic acid

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Lu X Y Barsh G S Akil H et al. Interaction between α-melanocyte-stimulating hormone and corticotropin-releasing hormone in the regulation of feeding and hypothalamo-pituitary-adrenal responses[J]. Journal of Neuroscience the Official Journal of the Society for Neuroscience 2003 23(21):7863.
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