CDK9-IN-2
CAS No. 1269815-17-9
CDK9-IN-2 ( CDK9 inhibitor II )
Catalog No. M11131 CAS No. 1269815-17-9
CDK9-IN-2 is a potent and selective CDK9 inhibitor with IC50 of <8 nM, example 4 in patent WO2011026917A1.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 76 | Get Quote |
|
5MG | 140 | Get Quote |
|
10MG | 223 | Get Quote |
|
25MG | 429 | Get Quote |
|
50MG | 628 | Get Quote |
|
100MG | 888 | Get Quote |
|
500MG | 1782 | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameCDK9-IN-2
-
NoteResearch use only, not for human use.
-
Brief DescriptionCDK9-IN-2 is a potent and selective CDK9 inhibitor with IC50 of <8 nM, example 4 in patent WO2011026917A1.
-
DescriptionCDK9-IN-2 is a potent and selective CDK9 inhibitor with IC50 of <8 nM, example 4 in patent WO2011026917A1.
-
SynonymsCDK9 inhibitor II
-
PathwayAngiogenesis
-
TargetCDK
-
RecptorCDK
-
Research AreaCancer
-
Indication——
Chemical Information
-
CAS Number1269815-17-9
-
Formula Weight363.81
-
Molecular FormulaC18H19ClFN3O2
-
Purity>98% (HPLC)
-
Solubility10 mM in DMSO
-
SMILESCOC1=C(C=C(C=C1)F)C2=CC(=NC=C2Cl)NC(=O)C3CCCNC3
-
Chemical Name3-Piperidinecarboxamide, N-[5-chloro-4-(5-fluoro-2-methoxyphenyl)-2-pyridinyl]-, (3R)-
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Keith B Pfister, et al. Heteroaryl compounds as kinase inhibitors. 2011, WO2011026917A1.
molnova catalog
related products
-
CDK5 inhibitor 20-22...
CDK5 inhibitor 20-223 (CP 668863) potent, selective, ATP-competitive CDK2/5 inhibitor with IC50 of 6.0 and 8.8 nM for CDK2/CyclinE and CDK5/p35, with little to no activity against CDK1/4/6/7/9.
-
FMF-04-159-2
FMF-04-159-2 is a potent, selective, covalent CDK14 inhibitor (IC50=86 nM) with pan-TAIRE family specificity (CDKs 14-18).
-
BAY 1251152
BAY 1251152 is the first potent, selective, orally available PTEFb/CDK9 inhibitor with biochemical IC50 of 9 nM and MOLM13 cell IC50 of 29 nM.