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Bupranolol

CAS No. 14556-46-8

Bupranolol( —— )

Catalog No. M22226 CAS No. 14556-46-8

Bupranolol is an antagonist of β2-adrenergic receptor,and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Bupranolol
  • Note
    Research use only, not for human use.
  • Brief Description
    Bupranolol is an antagonist of β2-adrenergic receptor,and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic.
  • Description
    Bupranolol is an antagonist of β2-adrenergic receptor，and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic.
  • In Vitro
    Bupranolol (1~3 μM) shifts isoprenaline-induced relaxation in the presence of 30 μM propranolol. Bupranolol acts as a competitive antagonist of isoprenaline-induced relaxation in the presence of 300 nM propranolol, with a pA2 value of 5.90. Bupranolol antagonizes β1- and β2-ARs with pA2 values of ≈9.0, and also antagonizes β3-AR with a pA2 value of 6.0.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    Adrenergic Receptor
  • Recptor
    β2-adrenergic receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    14556-46-8
  • Formula Weight
    271.78
  • Molecular Formula
    C14H22ClNO2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 50 mg/mL (183.97 mM)
  • SMILES
    OC(COC1=C(Cl)C=CC(C)=C1)CNC(C)(C)C
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Malinowska B , Kie?-Kononowicz K , Flau K , et al. Atypical cardiostimulant β-adrenoceptor in the rat heart: stereoselective antagonism by bupranolol but lack of effect by some bupranolol analogues[J]. 2003, 139(8):1548-1554.
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