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Bupranolol
CAS No. 14556-46-8
Bupranolol( —— )
Catalog No. M22226 CAS No. 14556-46-8
Bupranolol is an antagonist of β2-adrenergic receptor,and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 170 | In Stock |
|
| 10MG | 255 | In Stock |
|
| 25MG | 515 | In Stock |
|
| 50MG | 734 | In Stock |
|
| 100MG | 972 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBupranolol
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NoteResearch use only, not for human use.
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Brief DescriptionBupranolol is an antagonist of β2-adrenergic receptor,and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic.
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DescriptionBupranolol is an antagonist of β2-adrenergic receptor，and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic.
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In VitroBupranolol (1~3 μM) shifts isoprenaline-induced relaxation in the presence of 30 μM propranolol. Bupranolol acts as a competitive antagonist of isoprenaline-induced relaxation in the presence of 300 nM propranolol, with a pA2 value of 5.90. Bupranolol antagonizes β1- and β2-ARs with pA2 values of ≈9.0, and also antagonizes β3-AR with a pA2 value of 6.0.
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetAdrenergic Receptor
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Recptorβ2-adrenergic receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number14556-46-8
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Formula Weight271.78
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Molecular FormulaC14H22ClNO2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 50 mg/mL (183.97 mM)
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SMILESOC(COC1=C(Cl)C=CC(C)=C1)CNC(C)(C)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Malinowska B , Kie?-Kononowicz K , Flau K , et al. Atypical cardiostimulant β-adrenoceptor in the rat heart: stereoselective antagonism by bupranolol but lack of effect by some bupranolol analogues[J]. 2003, 139(8):1548-1554.
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