BRD32048
CAS No. 433694-46-3
BRD32048( BRD-32048 | BRD 32048 )
Catalog No. M27757 CAS No. 433694-46-3
BRD32048 is a top candidate ETV1 perturbagen. BRD32048 inhibits p300-dependent acetylation of ETV1, thereby promoting its degradation.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 155 | Get Quote |
|
10MG | 259 | Get Quote |
|
25MG | 484 | Get Quote |
|
50MG | 699 | Get Quote |
|
100MG | 981 | Get Quote |
|
200MG | Get Quote | Get Quote |
|
500MG | Get Quote | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
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Product NameBRD32048
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NoteResearch use only, not for human use.
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Brief DescriptionBRD32048 is a top candidate ETV1 perturbagen. BRD32048 inhibits p300-dependent acetylation of ETV1, thereby promoting its degradation.
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DescriptionBRD32048 is a top candidate ETV1 perturbagen. BRD32048 inhibits p300-dependent acetylation of ETV1, thereby promoting its degradation.
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In Vitro——
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In Vivo——
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SynonymsBRD-32048 | BRD 32048
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PathwayCell Cycle/DNA Damage
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TargetDNA/RNA Synthesis
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RecptorTEAD,YAP1/TAZ
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Research Area——
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Indication——
Chemical Information
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CAS Number433694-46-3
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Formula Weight314.393
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Molecular FormulaC16H22N6O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (397.60 mM)
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SMILESCOc1ccc(cc1)\N=c1/nc(CN2CCCCC2)nc(N)[nH]1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Ayumi Kaneda, et al. The novel potent TEAD inhibitor, K-975, inhibits YAP1/TAZ-TEAD protein-protein interactions and exerts an anti-tumor effect on malignant pleural mesothelioma. Am J Cancer Res. 2020 Dec 1;10(12):4399-4415.
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