BRD32048

CAS No. 433694-46-3

BRD32048( BRD-32048 | BRD 32048 )

Catalog No. M27757 CAS No. 433694-46-3

BRD32048 is a top candidate ETV1 perturbagen. BRD32048 inhibits p300-dependent acetylation of ETV1, thereby promoting its degradation.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 155 Get Quote
10MG 259 Get Quote
25MG 484 Get Quote
50MG 699 Get Quote
100MG 981 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    BRD32048
  • Note
    Research use only, not for human use.
  • Brief Description
    BRD32048 is a top candidate ETV1 perturbagen. BRD32048 inhibits p300-dependent acetylation of ETV1, thereby promoting its degradation.
  • Description
    BRD32048 is a top candidate ETV1 perturbagen. BRD32048 inhibits p300-dependent acetylation of ETV1, thereby promoting its degradation.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    BRD-32048 | BRD 32048
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    DNA/RNA Synthesis
  • Recptor
    TEAD,YAP1/TAZ
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    433694-46-3
  • Formula Weight
    314.393
  • Molecular Formula
    C16H22N6O
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 125 mg/mL (397.60 mM)
  • SMILES
    COc1ccc(cc1)\N=c1/nc(CN2CCCCC2)nc(N)[nH]1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Ayumi Kaneda, et al. The novel potent TEAD inhibitor, K-975, inhibits YAP1/TAZ-TEAD protein-protein interactions and exerts an anti-tumor effect on malignant pleural mesothelioma. Am J Cancer Res. 2020 Dec 1;10(12):4399-4415.
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