BRD-IN-26
CAS No. 1915012-19-9
BRD-IN-26 ( —— )
Catalog No. M13002 CAS No. 1915012-19-9
BRD-IN-26 is a potent bromodomain inhibitor that binds the fifth bromodomain of PB1 with a KD of 124 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
100MG | Get Quote | Get Quote |
|
200MG | Get Quote | Get Quote |
|
500MG | Get Quote | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameBRD-IN-26
-
NoteResearch use only, not for human use.
-
Brief DescriptionBRD-IN-26 is a potent bromodomain inhibitor that binds the fifth bromodomain of PB1 with a KD of 124 nM.
-
DescriptionBRD-IN-26 is a potent bromodomain inhibitor that binds the fifth bromodomain of PB1 with a KD of 124 nM, SMARCA2B and SMARCA4 with KD values of 262 and 417 nM, respectively; displays excellent selectivity over other bromodomains.
-
Synonyms——
-
PathwayChromatin/Epigenetic
-
TargetBromodomain
-
RecptorBromodomain
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number1915012-19-9
-
Formula Weight330.82
-
Molecular FormulaC17H19ClN4O
-
Purity>98% (HPLC)
-
Solubility——
-
SMILES——
-
Chemical Name(E)-6-chloro-3-((4-methylpiperazin-1-yl)methylene)-2,3-dihydropyrrolo[1,2-a]quinazolin-5(1H)-one
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Sutherell CL, et al. J Med Chem. 2016 May 26;59(10):5095-101.
molnova catalog
related products
-
CPI 0610
CPI 0610 is a potent, selective, and cell-active BET bromodomain inhibitor with IC50 of 39 nM for BRD4-BD1 in TR-FRET assay.
-
CPI-268456
A bromodomain-containing protein inhibitor.
-
GNE-781
GNE-781 (GNE781) is a potent, selective, non-CNS penetrant, orally active CBP/p300 bromodomain inhibitor.