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BRD-IN-26
CAS No. 1915012-19-9
BRD-IN-26 ( —— )
Catalog No. M13002 CAS No. 1915012-19-9
BRD-IN-26 is a potent bromodomain inhibitor that binds the fifth bromodomain of PB1 with a KD of 124 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameBRD-IN-26
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NoteResearch use only, not for human use.
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Brief DescriptionBRD-IN-26 is a potent bromodomain inhibitor that binds the fifth bromodomain of PB1 with a KD of 124 nM.
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DescriptionBRD-IN-26 is a potent bromodomain inhibitor that binds the fifth bromodomain of PB1 with a KD of 124 nM, SMARCA2B and SMARCA4 with KD values of 262 and 417 nM, respectively; displays excellent selectivity over other bromodomains.
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetBromodomain
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RecptorBromodomain
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Research Area——
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Indication——
Chemical Information
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CAS Number1915012-19-9
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Formula Weight330.82
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Molecular FormulaC17H19ClN4O
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name(E)-6-chloro-3-((4-methylpiperazin-1-yl)methylene)-2,3-dihydropyrrolo[1,2-a]quinazolin-5(1H)-one
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Sutherell CL, et al. J Med Chem. 2016 May 26;59(10):5095-101.
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