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BPN14770
CAS No. 1606974-33-7
BPN14770 ( —— )
Catalog No. M23705 CAS No. 1606974-33-7
BPN14770 is an allosteric inhibitor of selective phosphodiesterase 4D (PDE4D; IC50s: 7.8 nM and 7.4 nM for PDE4D7 and PDE4D3).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 205 | In Stock |
|
| 10MG | 385 | In Stock |
|
| 25MG | 644 | In Stock |
|
| 50MG | 888 | In Stock |
|
| 100MG | 1233 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBPN14770
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NoteResearch use only, not for human use.
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Brief DescriptionBPN14770 is an allosteric inhibitor of selective phosphodiesterase 4D (PDE4D; IC50s: 7.8 nM and 7.4 nM for PDE4D7 and PDE4D3).
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DescriptionBPN14770 is an allosteric inhibitor of selective phosphodiesterase 4D (PDE4D; IC50s: 7.8 nM and 7.4 nM for PDE4D7 and PDE4D3).
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorPDE4D3;PDE4D7
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Research Area——
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Indication——
Chemical Information
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CAS Number1606974-33-7
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Formula Weight405.8
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Molecular FormulaC21H15ClF3NO2
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Purity>98% (HPLC)
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SolubilityDMSO:260 mg/mL (640.71 mM; Need ultrasonic)
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SMILESOC(Cc1ccc(Cc2cc(-c3cccc(Cl)c3)nc(C(F)(F)F)c2)cc1)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Ricciarelli R, et al. Memory-enhancing effects of GEBR-32a, a new PDE4D inhibitor holding promise for the treatment of Alzheimer's disease. Sci Rep. 2017 Apr 12;7:46320.
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