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BI-1347
CAS No. 2163056-91-3
BI-1347 ( BI1347 )
Catalog No. M13451 CAS No. 2163056-91-3
BI-1347 is a potent, selective inhibitor of CDK8/cyclinC with IC50 of 1 nM。
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 72 | In Stock |
|
| 10MG | 115 | In Stock |
|
| 25MG | 228 | In Stock |
|
| 50MG | 417 | In Stock |
|
| 100MG | 614 | In Stock |
|
| 500MG | 1287 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBI-1347
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NoteResearch use only, not for human use.
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Brief DescriptionBI-1347 is a potent, selective inhibitor of CDK8/cyclinC with IC50 of 1 nM。
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DescriptionBI-1347 is a potent, selective inhibitor of CDK8/cyclinC with IC50 of 1 nM; BI-1347 shows tumor growth inhibition in an in vivo xenograft model, BI-1347 is an excellent small molecule tool inhibitor for testing biological hypotheses in vitro and in vivo.
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SynonymsBI1347
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PathwayAngiogenesis
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TargetCDK
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RecptorCDK8
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Research Area——
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Indication——
Chemical Information
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CAS Number2163056-91-3
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Formula Weight356.43
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Molecular FormulaC22H20N4O
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Purity>98% (HPLC)
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SolubilityDMSO: 120 mg/mL (336.68 mM), Need ultrasonic and warming （ < 1 mg/ml refers to the product slightly soluble or insoluble )
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SMILESO=C(N(C)C)CN1N=CC(C2=CC=C(C3=CN=CC4=C3C=CC=C4)C=C2)=C1
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Chemical Name2-(4-(4-(isoquinolin-4-yl)phenyl)-1H-pyrazol-1-yl)-N,N-dimethylacetamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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