BAY-6035

CAS No. 2247890-13-5

BAY-6035 ( BAY6035 )

Catalog No. M13611 CAS No. 2247890-13-5

BAY-6035 is a potent, peptide-competitive inhibitor of histone methyltransferase SMYD3.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 72 Get Quote
10MG 115 Get Quote
25MG 237 Get Quote
50MG 385 Get Quote
100MG 575 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    BAY-6035
  • Note
    Research use only, not for human use.
  • Brief Description
    BAY-6035 is a potent, peptide-competitive inhibitor of histone methyltransferase SMYD3.
  • Description
    BAY-6035 is a potent, peptide-competitive inhibitor of histone methyltransferase SMYD3, inhibits inhibits in vitro methylation of MEKK2 peptide with IC50 of 88 nM, >100-fold selectivity over other HMTases; inhibits the methylation of MEKK2 in cells with IC50 of 70 nM.
  • Synonyms
    BAY6035
  • Pathway
    Chromatin/Epigenetic
  • Target
    HMTase
  • Recptor
    HMTase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2247890-13-5
  • Formula Weight
    396.49
  • Molecular Formula
    C22H28N4O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C(C1=CC=C(N(C(N2CC3CC3C2)=O)[C@@H](C)CC(N4)=O)C4=C1)NCCC5CC5
  • Chemical Name
    (2S)-1-(3-azabicyclo[3.1.0]hexane-3-carbonyl)-N-(2-cyclopropylethyl)-2-methyl-4-oxo-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepine-7-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

molnova catalog
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