Atipamezole

CAS No. 104054-27-5

Atipamezole ( MPV-1248;MPV1248;MPV 1248 )

Catalog No. M10207 CAS No. 104054-27-5

Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 43 Get Quote
10MG 61 Get Quote
25MG 129 Get Quote
50MG 227 Get Quote
100MG 340 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    Atipamezole
  • Note
    Research use only, not for human use.
  • Brief Description
    Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM.
  • Description
    Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM; reverses the effects of the sedative dexmedetomidine and medetomidine as a veterinary drug.Alcoholism Phase 1 Discontinued
  • Synonyms
    MPV-1248;MPV1248;MPV 1248
  • Pathway
    Angiogenesis
  • Target
    Adrenergic Receptor
  • Recptor
    α2-adrenoceptor
  • Research Area
    Neurological Disease
  • Indication
    Alcoholism

Chemical Information

  • CAS Number
    104054-27-5
  • Formula Weight
    212.29
  • Molecular Formula
    C14H16N2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: ≥30 mg/mL
  • SMILES
    CCC1(C2=CNC=N2)CC3=C(C=CC=C3)C1
  • Chemical Name
    1H-Imidazole, 5-(2-ethyl-2,3-dihydro-1H-inden-2-yl)-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Pertovaara A, et al. CNS Drug Rev. 2005 Autumn;11(3):273-88.
2. Scheinin H, et al. Eur J Pharmacol. 1988 Jun 22;151(1):35-42.
3. Scheinin H, et al. Eur J Pharmacol. 1986 Sep 23;129(1-2):113-21.
4. Karhuvaara S, et al. Br J Clin Pharmacol. 1990 Jul;30(1):97-106.
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