Astemizole

CAS No. 68844-77-9

Astemizole ( NSC 329963 )

Catalog No. M15631 CAS No. 68844-77-9

Antihistamine drug now withdrawn from the market in many countries because of rare but potentially fatal side effects.

Purity : >98%(HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 38 In Stock
10MG 52 In Stock
25MG 85 In Stock
100MG Get Quote In Stock
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Biological Information

  • Product Name
    Astemizole
  • Note
    Research use only, not for human use.
  • Brief Description
    Antihistamine drug now withdrawn from the market in many countries because of rare but potentially fatal side effects.
  • Description
    Antihistamine drug now withdrawn from the market in many countries because of rare but potentially fatal side effects.
  • Synonyms
    NSC 329963
  • Pathway
    GPCR/G Protein
  • Target
    Histamine Receptor
  • Recptor
    H1 receptor; Potassium Channel
  • Research Area
    Inflammation/Immunology
  • Indication
    ——

Chemical Information

  • CAS Number
    68844-77-9
  • Formula Weight
    458.58
  • Molecular Formula
    C28H31FN4O
  • Purity
    >98%(HPLC)
  • Solubility
    Water: 432 mg/L
  • SMILES
    COC1=CC=C(C=C1)CCN2CCC(CC2)NC3=NC4=CC=CC=C4N3CC5=CC=C(C=C5)F
  • Chemical Name
    1-[(4-fluorophenyl)methyl]-N-[1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl]benzimidazol-2-amine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Salata JJ, et al. Circ Res. 1995 Jan;76(1):110-9.
molnova catalog
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