Aprocitentan
CAS No. 1103522-45-7
Aprocitentan ( ACT-132577 )
Catalog No. M21083 CAS No. 1103522-45-7
Aprocitentan is ETA and ETB antagonist .
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 222 | Get Quote |
|
10MG | 335 | Get Quote |
|
25MG | 566 | Get Quote |
|
50MG | 806 | Get Quote |
|
100MG | 1098 | Get Quote |
|
500MG | 2205 | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameAprocitentan
-
NoteResearch use only not for human use.
-
Brief DescriptionAprocitentan is ETA and ETB antagonist .
-
DescriptionAprocitentan is ETA and ETB antagonist .
-
SynonymsACT-132577
-
PathwayProteasome/Ubiquitin
-
TargetEndogenous Metabolite
-
RecptorET-A ;ET-B
-
Research AreaCardiovascular Disease
-
IndicationResistant Hypertension
Chemical Information
-
CAS Number1103522-45-7
-
Formula Weight546.19
-
Molecular FormulaC16H14Br2N6O4S
-
Purity>98% (HPLC)
-
SolubilityDMSO:46 mg/mL (84.22 mM)
-
SMILESNS(=O)(=O)Nc1ncnc(OCCOc2ncc(Br)cn2)c1-c1ccc(Br)cc1
-
Chemical NameN-[5-(4-bromophenyl)-6-{2-[(5-bromopyrimidin-2-yl)oxy]ethoxy}pyrimidin-4-yl]sulfuric diamide
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Trensz F Bortolamiol C Kramberg M et al. Journal of Pharmacology & Experimental Therapeutics 2019.
molnova catalog
related products
-
Phosphocholine chlor...
Phosphorylcholine is a small haptenic molecule is found in a wide variety of organisms. Human hepatic tumors undergo an elevation in the concentration of phosphorylcholine as the principal metabolic change is observed .
-
5-Aminovaleric acid
5-aminovalerate (or 5-aminopentanoic acid) is a lysine degradation product. It can be produced both endogenously or through bacterial catabolism of lysine.
-
L-(+)-Arabinose
L-(+)-Arabinose inhibits intestinal sucrase activity, thereby reducing sucrose utilization, and consequently decreasing lipogenesis.