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Antihistamine-1

CAS No. 1186430-60-3

Antihistamine-1 ( —— )

Catalog No. M26056 CAS No. 1186430-60-3

Antihistamine-1 is an H1-antihistamine (Ki: 6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel (IC50s: 5.4 and 0.8 μM).

Purity : >98% (HPLC)

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Datasheet

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Size	Price / USD	Stock	Quantity
5MG	80	Get Quote
10MG	140	Get Quote
25MG	281	Get Quote
50MG	529	Get Quote
100MG	759	Get Quote
200MG	Get Quote	Get Quote
500MG	Get Quote	Get Quote
1G	Get Quote	Get Quote

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Biological Information

Product Name

Antihistamine-1
Note

Research use only, not for human use.
Brief Description

Antihistamine-1 is an H1-antihistamine (Ki: 6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel (IC50s: 5.4 and 0.8 μM).
Description

Antihistamine-1 is an H1-antihistamine (Ki: 6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel (IC50s: 5.4 and 0.8 μM).(In Vitro):Antihistamine-1 is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively.
Synonyms

——
Pathway

Metabolic Enzyme/Protease
Target

P450
Recptor

——
Research Area

——
Indication

——

Chemical Information

CAS Number

1186430-60-3
Formula Weight

389.5
Molecular Formula

C23H24FN5
Purity

>98% (HPLC)
Solubility

——
SMILES

Cc1cnn(c1)C1CCN(CC1)c1nc2ccccc2n1Cc1ccc(F)cc1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

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