Aleplasinin

CAS No. 481629-87-2

Aleplasinin( PAZ-417 | PAZ 417 | PAZ417 )

Catalog No. M27948 CAS No. 481629-87-2

Aleplasinin is a selective and orally active inhibitor of Plasminogen activator inhibitor-1(PAI-1) and a key negative regulator of the fibrinolytic system. Aleplasinin can be used in Alzheimer's disease studies.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 135 In Stock
5MG 117 In Stock
10MG 188 In Stock
25MG 432 In Stock
50MG 641 In Stock
100MG 1014 In Stock
200MG 1358 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Aleplasinin
  • Note
    Research use only, not for human use.
  • Brief Description
    Aleplasinin is a selective and orally active inhibitor of Plasminogen activator inhibitor-1(PAI-1) and a key negative regulator of the fibrinolytic system. Aleplasinin can be used in Alzheimer's disease studies.
  • Description
    Aleplasinin is a selective and orally active inhibitor of Plasminogen activator inhibitor-1(PAI-1) and a key negative regulator of the fibrinolytic system. Aleplasinin can be used in Alzheimer's disease studies.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    PAZ-417 | PAZ 417 | PAZ417
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    PAI-1
  • Recptor
    nAChR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    481629-87-2
  • Formula Weight
    425.528
  • Molecular Formula
    C28H27NO3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 250 mg/mL (587.52 mM)
  • SMILES
    Cc1cccc(c1)-c1ccc2n(Cc3ccc(cc3)C(C)(C)C)cc(C(=O)C(O)=O)c2c1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Kimura I, et al. Inotropic effects of (+/-)-higenamine and its chemically related components, (+)-R-coclaurine and (+)-S-reticuline, contained in the traditional sino-Japanese medicines "bushi" and "shin-i" in isolated guinea pig papillary muscle. Jpn J Pharmacol. 1989 May;50(1):75-8.
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