Aleplasinin

CAS No. 481629-87-2

Aleplasinin( PAZ-417 | PAZ 417 | PAZ417 )

Catalog No. M27948 CAS No. 481629-87-2

Aleplasinin is a selective and orally active inhibitor of Plasminogen activator inhibitor-1(PAI-1) and a key negative regulator of the fibrinolytic system. Aleplasinin can be used in Alzheimer's disease studies.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 282 Get Quote
10MG 462 Get Quote
25MG 753 Get Quote
50MG 1044 Get Quote
100MG 1404 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    Aleplasinin
  • Note
    Research use only, not for human use.
  • Brief Description
    Aleplasinin is a selective and orally active inhibitor of Plasminogen activator inhibitor-1(PAI-1) and a key negative regulator of the fibrinolytic system. Aleplasinin can be used in Alzheimer's disease studies.
  • Description
    Aleplasinin is a selective and orally active inhibitor of Plasminogen activator inhibitor-1(PAI-1) and a key negative regulator of the fibrinolytic system. Aleplasinin can be used in Alzheimer's disease studies.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    PAZ-417 | PAZ 417 | PAZ417
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    PAI-1
  • Recptor
    nAChR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    481629-87-2
  • Formula Weight
    425.528
  • Molecular Formula
    C28H27NO3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 250 mg/mL (587.52 mM)
  • SMILES
    Cc1cccc(c1)-c1ccc2n(Cc3ccc(cc3)C(C)(C)C)cc(C(=O)C(O)=O)c2c1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Kimura I, et al. Inotropic effects of (+/-)-higenamine and its chemically related components, (+)-R-coclaurine and (+)-S-reticuline, contained in the traditional sino-Japanese medicines "bushi" and "shin-i" in isolated guinea pig papillary muscle. Jpn J Pharmacol. 1989 May;50(1):75-8.
molnova catalog
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