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AM-0902
CAS No. 1883711-97-4
AM-0902 ( —— )
Catalog No. M21665 CAS No. 1883711-97-4
AM-0902 is a potent and specific TRPA1 antagonist (IC50s: 71/131 nM for rTRPA1 and hTRPA1).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 69 | In Stock |
|
| 10MG | 96 | In Stock |
|
| 25MG | 200 | In Stock |
|
| 50MG | 389 | In Stock |
|
| 100MG | 575 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameAM-0902
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NoteResearch use only not for human use.
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Brief DescriptionAM-0902 is a potent and specific TRPA1 antagonist (IC50s: 71/131 nM for rTRPA1 and hTRPA1).
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DescriptionAM-0902 is a potent and specific TRPA1 antagonist (IC50s: 71/131 nM for rTRPA1 and hTRPA1).
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetTRP/TRPV Channel
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RecptorTRPA1
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Research Area——
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Indication——
Chemical Information
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CAS Number1883711-97-4
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Formula Weight370.79
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Molecular FormulaC17H15ClN6O2
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Purity>98% (HPLC)
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SolubilityDMSO: 145 mg/mL (391.05 mM; Need ultrasonic and warming)
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SMILESCn(cn1)c2c1N=CN(Cc1nc(CCc(cc3)ccc3Cl)no1)C2=O
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Chemical Name1-((3-(4-chlorophenethyl)-124-oxadiazol-5-yl)methyl)-7-methyl-17-dihydro-6H-purin-6-one
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Schenkel LB et al. Optimization of a Novel Quinazolinone-Based Series of Transient Receptor Potential A1 (TRPA1)Antagonists Demonstrating Potent in Vivo Activity. J Med Chem. 2016 Mar 24;59(6):2794-809.
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