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ACG-416B
CAS No. 95316-15-3
ACG-416B( ACG 416B )
Catalog No. M16812 CAS No. 95316-15-3
A potent, selective choline kinase α (ChoKα) inhibitor with IC50 of 0.13 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameACG-416B
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, selective choline kinase α (ChoKα) inhibitor with IC50 of 0.13 uM.
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DescriptionA potent, selective choline kinase α (ChoKα) inhibitor with IC50 of 0.13 uM, >385-fold selectivity over ChoKβ; demonstrates in vitro antiproliferative activity against HT29 cells with IC50 of 1.94 uM.
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In Vitro——
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In Vivo——
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SynonymsACG 416B
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PathwayOthers
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TargetChoK
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RecptorChoK
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Research Area——
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Indication——
Chemical Information
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CAS Number95316-15-3
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Formula Weight708.542
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Molecular FormulaC38H36Br2N4
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name1,1'-([1,1'-biphenyl]-3,3'-diylbis(methylene))bis(4-(methyl(phenyl)amino)pyridin-1-ium) bromide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Lacal JC, et al. Mol Cancer Ther. 2015 Jan;14(1):31-9.
2. Patent US 20110178124 A1. Pyridinium and quinolinium derivatives.
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