AC-262536
CAS No. 870888-46-3
AC-262536 ( AC 262536; AC262536 )
Catalog No. M27843 CAS No. 870888-46-3
AC-262536 is a selective androgen receptor (SAR) modulator and exhibits potent agonist activity at the androgen receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 35 | Get Quote |
|
5MG | 58 | Get Quote |
|
10MG | 102 | Get Quote |
|
25MG | 222 | Get Quote |
|
50MG | 380 | Get Quote |
|
100MG | 565 | Get Quote |
|
500MG | 1215 | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
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Product NameAC-262536
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NoteResearch use only, not for human use.
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Brief DescriptionAC-262536 is a selective androgen receptor (SAR) modulator and exhibits potent agonist activity at the androgen receptor.
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DescriptionAC-262536 is a selective androgen receptor (SAR) modulator and exhibits potent agonist activity at the androgen receptor. It has partial agonist activity with respect to testosterone and suppresses luteinizing hormone.(In Vitro):AC-262536 inhibits dihydroxytestosterone (DHT)-induced proliferation of LNCaP in a dose-dependent manner. The effects are significant with 100 nM, and reaches a plateau with 1 μM.(In Vivo):In male sprague-dawley rats, administration of AC-262536 (subcutaneous injection, once daily for 14 consecutive days) significantly decreased LH levels by about 40% at the 3 mg/kg dose. At the 10 and 30 mg/kg doses, the effects of AC-262536 were significantly stronger than Testosterone Propionate (TP) : 1.91±0.32 ng/mL and 1.53±0.34 ng/mL vs. 3.12±0.69 ng/mL, respectively.
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SynonymsAC 262536; AC262536
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PathwayEndocrinology/Hormones
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TargetAndrogen Receptor (AR)
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number870888-46-3
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Formula Weight278.4
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Molecular FormulaC18H18N2O
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Purity>98% (HPLC)
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Solubility——
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SMILESOC1C[C@@H]2CC[C@H](C1)N2c1ccc(C#N)c2ccccc12
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.El-Sayed, May A.; Al-Gendy, Amal. A.; Hamdan, Dalia. I.; El-Shazly, Assem M. Phytoconstituents, LC-?ESI-?MS profile, antioxidant and antimicrobial activities of Citrus x limon L. Burm. f. Cultivar variegated pink lemon. Journal of Pharmaceutical Sciences and Research (2017), 9(4), 375-391.
molnova catalog
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