1NM-PP1
CAS No. 221244-14-0
1NM-PP1 ( PP1 Analog II )
Catalog No. M13527 CAS No. 221244-14-0
1NM-PP1(PP1 Analog II) is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors(IC50=28 uM vSrc; 4.2 nM v-Src-as1 I338G).
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 54 | In Stock |
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5MG | 73 | In Stock |
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10MG | 128 | In Stock |
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25MG | 272 | In Stock |
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50MG | 504 | In Stock |
|
100MG | 669 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
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Biological Information
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Product Name1NM-PP1
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NoteResearch use only, not for human use.
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Brief Description1NM-PP1(PP1 Analog II) is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors(IC50=28 uM vSrc; 4.2 nM v-Src-as1 I338G).
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Description1NM-PP1(PP1 Analog II) is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors(IC50=28 uM vSrc; 4.2 nM v-Src-as1 I338G).
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SynonymsPP1 Analog II
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PathwayAngiogenesis
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TargetCDK
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RecptorCDK7
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number221244-14-0
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Formula Weight331.41
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Molecular FormulaC20H21N5
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Purity>98%(HPLC)
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SolubilityDMSO: 10 mM
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SMILESNC1=C2C(N(C(C)(C)C)N=C2CC3=C4C=CC=CC4=CC=C3)=NC=N1
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Chemical Name1-(tert-butyl)-3-(naphthalen-1-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Papa FR, et al. Science. 2003 Nov 28;302(5650):1533-7.
molnova catalog
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