BML-259

CAS No. 267654-00-2

BML-259( CAY10554 )

Catalog No. M28107 CAS No. 267654-00-2

BML-259 is an inhibitor of CDK5 and CDK2 with IC50s of 64 and 98 nM, respectively. BML-259 can be used in studies about the treatment of cancer and neurodegenerative diseases.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 39 Get Quote
10MG 69 Get Quote
25MG 155 Get Quote
50MG 264 Get Quote
100MG 462 Get Quote
500MG 981 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    BML-259
  • Note
    Research use only, not for human use.
  • Brief Description
    BML-259 is an inhibitor of CDK5 and CDK2 with IC50s of 64 and 98 nM, respectively. BML-259 can be used in studies about the treatment of cancer and neurodegenerative diseases.
  • Description
    BML-259 is an inhibitor of CDK5 and CDK2 with IC50s of 64 and 98 nM, respectively. BML-259 can be used in studies about the treatment of cancer and neurodegenerative diseases.(In Vitro):BML-259 prevents a large population of cells from NAC-evoked cell death.
  • In Vitro
    BML-259 (10 μM) protects large population of cells against non-Aβ component of Alzheimer's disease amyloid (NAC)-evoked cell death.
  • In Vivo
    ——
  • Synonyms
    CAY10554
  • Pathway
    Angiogenesis
  • Target
    CDK
  • Recptor
    Antifungal|Antiviral
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    267654-00-2
  • Formula Weight
    260.36
  • Molecular Formula
    C14H16N2OS
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 125 mg/mL (480.12 mM)
  • SMILES
    O=C(NC1=NC=C(S1)C(C)C)CC=2C=CC=CC2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Freitas-Silva O, et al. Tracing fungi secondary metabolites in Brazil nuts using LC-MS/MS. Drug Metab Lett. 2011 Aug;5(3):150-5.
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