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(3aR)-Selitrectinib
CAS No. 1350884-56-8
(3aR)-Selitrectinib( BAY 2731954 | (6RS)-LOXO-195 )
Catalog No. M28716 CAS No. 1350884-56-8
(6RS)-LOXO-195 is a potent and selective Trk tyrosine kinase inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 43 | Get Quote |
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| 5MG | 72 | Get Quote |
|
| 10MG | 110 | Get Quote |
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| 25MG | 215 | Get Quote |
|
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
|
Biological Information
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Product Name(3aR)-Selitrectinib
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NoteResearch use only, not for human use.
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Brief Description(6RS)-LOXO-195 is a potent and selective Trk tyrosine kinase inhibitor.
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Description(6RS)-LOXO-195 is a potent and selective Trk tyrosine kinase inhibitor.
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In Vitro——
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In Vivo——
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SynonymsBAY 2731954 | (6RS)-LOXO-195
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PathwayTyrosine Kinase
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TargetTrk Receptor
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RecptorApoptosis|MARK3|MARK4
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Research Area——
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Indication——
Chemical Information
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CAS Number1350884-56-8
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Formula Weight380.427
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Molecular FormulaC20H21FN6O
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Purity>98% (HPLC)
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Solubility——
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SMILES[H][C@]12CCCN1c1ccn3ncc(C(=O)NC(C)CCc4ncc(F)cc24)c3n1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Fangfang Li, et al. PCC0208017, a novel small-molecule inhibitor of MARK3/MARK4, suppresses glioma progression?in vitro?and?in vivo. Acta Pharm Sin B.2020 Feb;10(2):289-300.
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