YM976

CAS No. 191219-80-4

YM976 ( —— )

Catalog No. M21141 CAS No. 191219-80-4

YM976 is an orally active PDE4 inhibitor (IC50:2.2 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 39 Get Quote
10MG 63 Get Quote
25MG 104 Get Quote
100MG Get Quote Get Quote
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Biological Information

  • Product Name
    YM976
  • Note
    Research use only not for human use.
  • Brief Description
    YM976 is an orally active PDE4 inhibitor (IC50:2.2 nM).
  • Description
    YM976 is an orally active PDE4 inhibitor (IC50:2.2 nM).
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    PDE
  • Recptor
    PDE4
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    191219-80-4
  • Formula Weight
    313.78
  • Molecular Formula
    C17H16ClN3O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CCc1ccc2c(-c3cccc(Cl)c3)nc(=O)n(CC)c2n1
  • Chemical Name
    4-(3-chlorophenyl)-17-diethyl-1H2H-pyrido[23-d]pyrimidin-2-one

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Aoki M Kobayashi M Ishikawa J et al. A Novel Phosphodiesterase Type 4 Inhibitor YM976 (4-(3-Chlorophenyl)-17-diethylpyrido[23-d]pyrimidin-2(1H)-one) with Little Emetogenic Activity[J]. Journal of Pharmacology & Experimental Therapeutics 2000 295(1):255-260.
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