XEN-907

CAS No. 912656-34-9

XEN-907 ( XEN907;XEN 907 )

Catalog No. M16553 CAS No. 912656-34-9

A potent, selective NaV1.7 blocker with IC50 of 3 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 57 Get Quote
5MG 87 Get Quote
10MG 129 Get Quote
25MG 214 Get Quote
50MG 322 Get Quote
100MG Get Quote Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    XEN-907
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent, selective NaV1.7 blocker with IC50 of 3 nM.
  • Description
    A potent, selective NaV1.7 blocker with IC50 of 3 nM; shows no significant activity at 10 uM against a broad panel of 63 receptors and transporters; has no cytotoxic and favourable hepatocyte metabolic stability for both human and dog,Pain Preclinical
  • Synonyms
    XEN907;XEN 907
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    Sodium Channel
  • Recptor
    Sodium Channel
  • Research Area
    Neurological Disease
  • Indication
    Pain

Chemical Information

  • CAS Number
    912656-34-9
  • Formula Weight
    351.40
  • Molecular Formula
    C21H21NO4
  • Purity
    >98% (HPLC)
  • Solubility
    10 mM in DMSO
  • SMILES
    O=C(C12COC3=C1C=C(OCO4)C4=C3)N(CCCCC)C5=C2C=CC=C5
  • Chemical Name
    Spiro[furo[2,3-f]-1,3-benzodioxole-7(6H),3'-[3H]indol]-2'(1'H)-one, 1'-pentyl-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Chowdhury S, et al. Bioorg Med Chem Lett. 2011 Jun 15;21(12):3676-81.
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