XEN-907
CAS No. 912656-34-9
XEN-907 ( XEN907;XEN 907 )
Catalog No. M16553 CAS No. 912656-34-9
A potent, selective NaV1.7 blocker with IC50 of 3 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 57 | Get Quote |
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5MG | 87 | Get Quote |
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10MG | 129 | Get Quote |
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25MG | 214 | Get Quote |
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50MG | 322 | Get Quote |
|
100MG | Get Quote | Get Quote |
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200MG | Get Quote | Get Quote |
|
500MG | Get Quote | Get Quote |
|
1G | Get Quote | Get Quote |
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Biological Information
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Product NameXEN-907
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, selective NaV1.7 blocker with IC50 of 3 nM.
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DescriptionA potent, selective NaV1.7 blocker with IC50 of 3 nM; shows no significant activity at 10 uM against a broad panel of 63 receptors and transporters; has no cytotoxic and favourable hepatocyte metabolic stability for both human and dog,Pain Preclinical
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SynonymsXEN907;XEN 907
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PathwayMembrane Transporter/Ion Channel
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TargetSodium Channel
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RecptorSodium Channel
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Research AreaNeurological Disease
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IndicationPain
Chemical Information
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CAS Number912656-34-9
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Formula Weight351.40
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Molecular FormulaC21H21NO4
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESO=C(C12COC3=C1C=C(OCO4)C4=C3)N(CCCCC)C5=C2C=CC=C5
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Chemical NameSpiro[furo[2,3-f]-1,3-benzodioxole-7(6H),3'-[3H]indol]-2'(1'H)-one, 1'-pentyl-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Chowdhury S, et al. Bioorg Med Chem Lett. 2011 Jun 15;21(12):3676-81.
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