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WZ4003
CAS No. 1214265-58-3
WZ4003 ( WZ4003; WZ-4003; WZ 4003 )
Catalog No. M10799 CAS No. 1214265-58-3
WZ4003 is a highly specific NUAK kinase inhibitor with IC50 of 20 nM and 100 nM for NUAK1 and NUAK2, respectively.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 39 | In Stock |
|
| 10MG | 63 | In Stock |
|
| 25MG | 107 | In Stock |
|
| 50MG | 160 | In Stock |
|
| 100MG | 241 | In Stock |
|
| 200MG | 357 | In Stock |
|
| 500MG | 590 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameWZ4003
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NoteResearch use only, not for human use.
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Brief DescriptionWZ4003 is a highly specific NUAK kinase inhibitor with IC50 of 20 nM and 100 nM for NUAK1 and NUAK2, respectively.
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DescriptionWZ4003 is a highly specific NUAK kinase inhibitor with IC50 of 20 nM and 100 nM for NUAK1 and NUAK2, respectively, without significant inhibition on 139 other kinases.
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SynonymsWZ4003; WZ-4003; WZ 4003
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PathwayMembrane Transporter/Ion Channel
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TargetAMPK
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RecptorNUAK1; NUAK2
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1214265-58-3
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Formula Weight496.99
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Molecular FormulaC25H29ClN6O3
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Purity>98%(HPLC)
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SolubilityDMSO:7 mg/mL (14.08 mM); Ethanol:<1 mg/mL (<1 mM); Water：<1 mg/mL (<1 mM)
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SMILESCCC(NC1=CC=CC(OC2=NC(NC3=CC=C(N4CCN(C)CC4)C=C3OC)=NC=C2Cl)=C1)=O
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Chemical NameN-[3-[[5-chloro-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-4-pyrimidinyl]oxy]phenyl]-propanamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Banerjee S, et al. Biochem J. 2014, 457(1), 215-225.
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