Cart
sales@molnova.com
Home - Products - Cell Cycle/DNA Damage - Potassium Channel - VU0810464

VU0810464

CAS No. 2126040-21-7

VU0810464 ( —— )

Catalog No. M21143 CAS No. 2126040-21-7

VU0810464 is a non-ureaG protein-gated inwardly-rectifying potassium channels (GIRK Kir3) activator.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 259 Get Quote
10MG 404 Get Quote
25MG 665 Get Quote
50MG 888 Get Quote
100MG 1251 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote
Group Booking Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    VU0810464
  • Note
    Research use only not for human use.
  • Brief Description
    VU0810464 is a non-ureaG protein-gated inwardly-rectifying potassium channels (GIRK Kir3) activator.
  • Description
    VU0810464 is a non-ureaG protein-gated inwardly-rectifying potassium channels (GIRK Kir3) activator.
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    Potassium Channel
  • Recptor
    GIRK
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2126040-21-7
  • Formula Weight
    349.83
  • Molecular Formula
    C18H21ClFN3O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:250 mg/mL (714.63 mM)
  • SMILES
    Cc1cc(NC(=O)Cc2ccc(F)c(Cl)c2)n(C2CCCCC2)n1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Discovery and Characterization of 1H?Pyrazol-5-yl-2-phenylacetamides as Novel Non-Urea-Containing GIRK1/2 Potassium Channel Activators[J]. Acs Chemical Neuroscience 2017 8(9):1873-1879.
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • Tertiapin-Q

    A high affinity blocker for inward-rectifier K+ channels, this compound is a stable derivative of the bee venom toxin tertiapin. Binds to ROMK1 (Kir1.1) and GIRK1/4 (Kir3.1/3.4) channels with high affinity (Ki values are 1.3 and 13.3 nM respectively) and is selective over Kir2.1 channels. Derivative tertiapin LQ also available.

  • DMP 543

    A potent blocker of voltage-gated potassium channels Kv7 (KCNQ) that enhances ACh release from rat hippocampal slices in vitro with EC50 of 0.7 uM.

  • NS11021

    NS11021, a novel opener of large-conductance Ca(2+)-activated K(+) channels.

Sign In Join Free