VU0238429
CAS No. 1160247-92-6
VU0238429 ( SCR-1481B1 )
Catalog No. M21562 CAS No. 1160247-92-6
VU0238429 is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 35 | Get Quote |
|
5MG | 58 | Get Quote |
|
10MG | 102 | Get Quote |
|
25MG | 205 | Get Quote |
|
50MG | 288 | Get Quote |
|
100MG | 507 | Get Quote |
|
200MG | Get Quote | Get Quote |
|
500MG | Get Quote | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameVU0238429
-
NoteResearch use only not for human use.
-
Brief DescriptionVU0238429 is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).
-
DescriptionVU0238429 is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).
-
SynonymsSCR-1481B1
-
PathwayEndocrinology/Hormones
-
TargetAChR
-
RecptorM5 mAChR
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number1160247-92-6
-
Formula Weight351.28
-
Molecular FormulaC17H12F3NO4
-
Purity>98% (HPLC)
-
SolubilityDMSO:150 mg/mL (427.01 mM)
-
SMILESCOc1ccc(CN2C(=O)C(=O)c3cc(OC(F)(F)F)ccc23)cc1
-
Chemical Name1-[(4-methoxyphenyl)methyl]-5-(trifluoromethoxy)-23-dihydro-1H-indole-23-dione
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Bridges TM et al. Discovery of the first highly M5-preferring muscarinic acetylcholine receptor ligand an M5 positive allosteric modulator derived from a series of 5-trifluoromethoxy N-benzyl isatins.
molnova catalog
related products
-
Pirenzepine dihydroc...
An antimuscarinic agent that inhibits gastric secretion at lower doses than are required to affect gastrointestinal motility, salivary, central nervous system, cardiovascular, ocular, and urinary function.
-
Clothianidin
Clothianidin, an insecticide, acts as an agonist of acetylcholine to stimulate nAChR, thereby activating post-synaptic acetylcholine receptors but not inhibiting AChE.
-
5-Hydroxy-1,7-diphen...
5-Hydroxy-1, 7-diphenyl-6-hepten-3-one has antioxidant activity.