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Home - Products - Endocrinology/Hormones - Androgen Receptor (AR) - VPC-13566

VPC-13566

CAS No. 218464-59-6

VPC-13566 ( VPC13566; VPC 13566 )

Catalog No. M27935 CAS No. 218464-59-6

VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the BF3 pocket.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 191 Get Quote
10MG 267 Get Quote
25MG 466 Get Quote
50MG 674 Get Quote
100MG 954 Get Quote
500MG 1881 Get Quote
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Biological Information

  • Product Name
    VPC-13566
  • Note
    Research use only, not for human use.
  • Brief Description
    VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the BF3 pocket.
  • Description
    VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the BF3 pocket. VPC-13566 inhibits the growth of various prostate cancer cell lines and reduces the growth of AR-dependent prostate cancer xenograft tumors in mice.
  • Synonyms
    VPC13566; VPC 13566
  • Pathway
    Endocrinology/Hormones
  • Target
    Androgen Receptor (AR)
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    218464-59-6
  • Formula Weight
    258.3
  • Molecular Formula
    C18H14N2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Cc1cccc2c(c[nH]c12)-c1ccc2ccccc2n1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Anthony Boitano, et al. Aryl hydrocarbon receptor antagonists and methods of use thereof for treating various diseases. WO2020051207A2
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