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VPC-13566

CAS No. 218464-59-6

VPC-13566( VPC13566 | VPC 13566 )

Catalog No. M27935 CAS No. 218464-59-6

VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the BF3 pocket.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 191 Get Quote
10MG 267 Get Quote
25MG 466 Get Quote
50MG 674 Get Quote
100MG 954 Get Quote
500MG 1881 Get Quote
1G Get Quote Get Quote
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Biological Information

  • Product Name
    VPC-13566
  • Note
    Research use only, not for human use.
  • Brief Description
    VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the BF3 pocket.
  • Description
    VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the BF3 pocket. VPC-13566 inhibits the growth of various prostate cancer cell lines and reduces the growth of AR-dependent prostate cancer xenograft tumors in mice.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    VPC13566 | VPC 13566
  • Pathway
    Endocrinology/Hormones
  • Target
    Androgen Receptor (AR)
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    218464-59-6
  • Formula Weight
    258.324
  • Molecular Formula
    C18H14N2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (387.12 mM)
  • SMILES
    Cc1cccc2c(c[nH]c12)-c1ccc2ccccc2n1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Anthony Boitano, et al. Aryl hydrocarbon receptor antagonists and methods of use thereof for treating various diseases. WO2020051207A2
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