UPCDC30245

CAS No. 1883351-01-6

UPCDC30245 ( UPCDC 30245 )

Catalog No. M12921 CAS No. 1883351-01-6

UPCDC30245 is an allosteric inhibitor of AAA ATPase p97 with IC50 of 27 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    UPCDC30245
  • Note
    Research use only, not for human use.
  • Brief Description
    UPCDC30245 is an allosteric inhibitor of AAA ATPase p97 with IC50 of 27 nM.
  • Description
    UPCDC30245 is an allosteric inhibitor of AAA ATPase p97 with IC50 of 27 nM, binds at the junction between the D1 and D2 domains of p97.
  • Synonyms
    UPCDC 30245
  • Pathway
    Proteasome/Ubiquitin
  • Target
    p97
  • Recptor
    p97
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1883351-01-6
  • Formula Weight
    463.63
  • Molecular Formula
    C28H38FN5
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CC(N1CCN(CCNC2CCN(C3=CC=CC(C(N4)=CC5=C4C=CC(F)=C5)=C3)CC2)CC1)C
  • Chemical Name
    1-(3-(5-Fluoro-1H-indol-2-yl)phenyl)-N-(2-(4-isopropylpiperazin-1-yl)ethyl)piperidin-4-amine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Segura-Cabrera A, et al. Sci Rep. 2017 Mar 21;7:44912.
2. Banerjee S, et al. Science. 2016 Feb 19;351(6275):871-5.
molnova catalog
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