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Tocainide
CAS No. 41708-72-9
Tocainide( —— )
Catalog No. M24378 CAS No. 41708-72-9
Tocainide is a blocker of the sodium channel and used for the treatment of tinnitus.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 76 | In Stock |
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| 5MG | 35 | In Stock |
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| 10MG | 58 | In Stock |
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| 25MG | 95 | In Stock |
|
| 50MG | 138 | In Stock |
|
| 100MG | 206 | In Stock |
|
| 500MG | 512 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTocainide
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NoteResearch use only, not for human use.
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Brief DescriptionTocainide is a blocker of the sodium channel and used for the treatment of tinnitus.
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DescriptionTocainide is a blocker of the sodium channel and used for the treatment of tinnitus.(In Vivo):Tocainide (100 mg/kg) effectively suppresses ventricular ectopic activity in unanesthetized dogs with coronary occlusion. Termination of tocainide infusion in both digitalis toxicity and coronary occlusion models results in prompt return of ventricular ectopic activity.
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In Vitro——
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In VivoTocainide (100 mg/kg) effectively suppresses ventricular ectopic activity in unanesthetized dogs with coronary occlusion. Termination of tocainide infusion in both digitalis toxicity and coronary occlusion models results in prompt return of ventricular ectopic activity.
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetSodium Channel
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Recptorsodium channel
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Research Area——
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Indication——
Chemical Information
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CAS Number41708-72-9
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Formula Weight192.13
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Molecular FormulaC11H16N2O
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Purity>98% (HPLC)
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SolubilityDMSO:10 mM
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SMILESCC(N)C(NC1=C(C)C=CC=C1C)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Alpert JS, et al. Chemistry, pharmacology, antiarrhythmic efficacy and adverse effects of tocainide hydrochloride, an orally active structural analog of lidocaine. Pharmacotherapy. 1983 Nov-Dec;3(6):316-23.
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